| Authors |
Yudhi D. Kurniawan, Kellie L. Tuck, Sergio Castillón, Andrea J. Robinson |
| Published | Tetrahedron Letters |
| Graphical abstract |  |
| Abstract |
A convergent synthesis of the C3-C8 fragment of zaragozic acids is described. The key reactions include desilylation-aldol reaction, rearrangement induced by regioselective reductive cleavage, BAIB/TEMPO-Pinnick oxidation, esterification, silylation, and hydrogenolysis. |
| Citation |
B. Zhang, B. H. Fraser, M. A. Klenner, Z. Chen, S. H. Liang, M Massi, A. J. Robinson, G. Pascali, “[ 18 F]Ethenesulfonyl Fluoride as a Practical Radiofluoride Relay Reagent”, Chemistry – A European Journal, 2019, 25(32), 7613-7617 |
| Doi | |
| Keywords |
Zaragozic acids |
-
Recent Posts
- Minimizing Mitogenic Potency of Insulin Analogues Through Modification of a Disulfide Bond
- Toward the stereoselective synthesis of zaragozic acid framework: A desilylation-aldol reaction approach
- [18 F]Ethenesulfonyl Fluoride as a Practical Radiofluoride Relay Reagent
- Bioinspired carrier-free peptide conjugated BF2-oxasmaragdyrin dye-based nano self-assemblies: a photostable NIR cancer theragnostic agent
- Design, Development, In Vitro and Preliminary In Vivo Evaluation of a Novel Photo-Angioplasty Device: Lumi-Solve
- BF2-Oxasmaragdyrin Nanoparticles: A Non-toxic, Photostable, Enhanced Non-radiative Decay-Assisted Efficient Photothermal Cancer Theragnostic Agent
- Synthesis and Studies of Glucosamine Conjugated BF2 -Oxasmaragdyrin
- Cell-Penetrating Peptide-Conjugated BF 2 -Oxasmaragdyrins as NIRF Imaging and Photothermal Agents”
Archives
Categories
Meta
Andrea Robinson Group 