-
Recent Posts
- Minimizing Mitogenic Potency of Insulin Analogues Through Modification of a Disulfide Bond
- Toward the stereoselective synthesis of zaragozic acid framework: A desilylation-aldol reaction approach
- [18 F]Ethenesulfonyl Fluoride as a Practical Radiofluoride Relay Reagent
- Bioinspired carrier-free peptide conjugated BF2-oxasmaragdyrin dye-based nano self-assemblies: a photostable NIR cancer theragnostic agent
- Design, Development, In Vitro and Preliminary In Vivo Evaluation of a Novel Photo-Angioplasty Device: Lumi-Solve
- BF2-Oxasmaragdyrin Nanoparticles: A Non-toxic, Photostable, Enhanced Non-radiative Decay-Assisted Efficient Photothermal Cancer Theragnostic Agent
- Synthesis and Studies of Glucosamine Conjugated BF2 -Oxasmaragdyrin
- Cell-Penetrating Peptide-Conjugated BF 2 -Oxasmaragdyrins as NIRF Imaging and Photothermal Agents”
Archives
Categories
Meta
Monthly Archives: September 2014
A Concise Cross-Metathesis Route to Enantiopure 1-Azaspirocycles
Authors Zhen James Wang, Nicolas Daniel Spiccia, Christopher James Gartshore, Jayamini Illesinghe, William Roy Jackson and Andrea Jane Robinson Published Synthesis Graphical abstract Abstract The 1-azaspirocyclic ring system can be found in a number of bioactive natural product families. … Continue reading →
Posted in Metathesis, Publications, Publications 2013
|
Tagged dicarba peptides, Metathesis
|
Leave a comment
Combinatorial Approach for the Rapid Determination of Thermochromic Behavior of Binary and Ternary Cholesteric Liquid Crystalline Mixtures
Authors Louise C. van der Werff, Andrea J. Robinson and Ilias L. Kyratzis Published ACS Combinatorial Science Graphical abstract Abstract A combinatorial approach was developed for the rapid determination of thermochromic behavior of a large number of binary and … Continue reading →
Posted in Fibres, Publications, Publications 2012
|
Tagged dicarba peptides, Metathesis
|
Leave a comment
A one pot, metathesis–hydrogenation sequence for the selective formation of carbon–carbon bonds
Authors Andrea J. Robinson, Jomana Elaridi, Jim Patel and W. Roy Jackson Published Chemical Communications Graphical abstract Abstract The selective formation of C–C bonds in complex molecules is one of the major challenges in organic chemistry. Olefin metathesis provides … Continue reading →
Posted in Dicarba peptides, Metathesis, Publications, Publications pre 2009
|
Tagged dicarba peptides, Metathesis
|
Leave a comment
Solid phase synthesis and structural analysis of novel A-chain dicarba analogs of human relaxin-3 (INSL7) that exhibit full biological activity
Authors Mohammed Akhter Hossain, K. Johan Rosengren, Suode Zhang, Ross A. D. Bathgate, Geoffrey W. Tregear, Bianca J. van Lierop, Andrea J. Robinson and John D. Wade Published Organic & Biomolecular Chemistry Graphical abstract Abstract Replacement of disulfide bonds … Continue reading →
Controlled Synthesis of (S,S)-2,7-Diaminosuberic Acid: A Method for Regioselective Construction of Dicarba Analogues of Multicystine-Containing Peptides
Authors Jomana Elaridi, Jim Patel, W. Roy Jackson and Andrea J. Robinson Published Journal of Organic Chemistry Graphical abstract Abstract A method to facilitate regioselective formation of multiple dicarba isosteres of cystine is described. A sequence of ruthenium-catalyzed cross … Continue reading →
Electrostatic immobilization of an olefin metathesis pre-catalyst on iron oxide magnetic particles
Authors Matthew J. Byrnes, Andrew M. Hilton, Clint P. Woodward, William R. Jackson and Andrea J. Robinson Published Green Chemistry Graphical abstract Abstract Homogenous Grubbs-type pre-catalysts have played an important role in the application of olefin metathesis to organic … Continue reading →
A simple amine protection strategy for olefin metathesis reactions
Authors Clint Peter Woodward, Nicolas Daniel Spiccia, William Roy Jackson and Andrea Jane Robinson Published Chemical Communications Graphical abstract Abstract Acyclic diamines are valuable feedstocks for polyamide synthesis. Ruthenium-alkylidene catalysed cross metathesis of amino alkenes is problematic and acyl … Continue reading →
Thermochromic composite fibres containing liquid crystals formed via melt extrusion
Authors Louise van der Werff, Ilias Louis Kyratzis, Andrea Robinson, Robin Cranston, Gary Peeters, Mike O’Shea and Lance Nichols Published Journal of Material Science Graphical abstract Abstract Temperature-sensitive fibres and textiles can be applied to a variety of medical … Continue reading →
Dicarba α‐Conotoxin Vc1.1 Analogues with Differential Selectivity for Nicotinic Acetylcholine and GABAB Receptors
Authors Bianca J. van Lierop, Samuel D. Robinson, Shiva N. Kompella, Alessia Belgi, Jeffrey R. McArthur, Andrew Hung, Christopher A. MacRaild, David J. Adams, Raymond S. Norton and Andrea J. Robinson Published ACS Chemical Biology Graphical abstract Abstract Conotoxins … Continue reading →
Posted in Conotoxins, Dicarba peptides, Metathesis, Publications, Publications 2013
|
Leave a comment
An Efficient Protocol for the Cross-Metathesis of Sterically Demanding Olefins
Authors Zhen J. Wang, W. Roy Jackson and Andrea J. Robinson Published Organic Letters Graphical abstract Abstract We have recently described synthetic routes to the azaspirocyclic ring systems found in marine tricyclic alkaloids such as Cylindricine A utilising a … Continue reading →
Andrea Robinson Group 