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Category Archives: Dicarba peptides
Stereoselective Synthesis and Structural Elucidation of Dicarba Peptides
Authors Ellen C. Gleeson, Zhen J. Wang, Samuel D. Robinson, Sandeep Chhabra, Christopher A. MacRaild, W. Roy Jackson, Raymond S. Norton and Andrea J. Robinson Published Chemical Communications Graphical abstract Abstract Preformed, orthogonally-protected Z– and E-diaminosuberic acid residues can be used to synthesise target dicarba peptides. … Continue reading →
A one-pot selective homodimerisation/hydrogenation strategy for sequential dicarba bridge formation
Authors James Burnley, W. Roy Jackson and Andrea J. Robinson Published Journal of Organic Chemistry Graphical abstract Abstract The installation of interlocked dicarba bridges into peptide sequences requires the development of regioselective and chemoselective methodology. This manuscript describes a one-pot, … Continue reading →
Posted in Dicarba peptides, Metathesis, Publications, Publications 2015
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A one pot, metathesis–hydrogenation sequence for the selective formation of carbon–carbon bonds
Authors Andrea J. Robinson, Jomana Elaridi, Jim Patel and W. Roy Jackson Published Chemical Communications Graphical abstract Abstract The selective formation of C–C bonds in complex molecules is one of the major challenges in organic chemistry. Olefin metathesis provides … Continue reading →
Posted in Dicarba peptides, Metathesis, Publications, Publications pre 2009
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Tagged dicarba peptides, Metathesis
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Solid phase synthesis and structural analysis of novel A-chain dicarba analogs of human relaxin-3 (INSL7) that exhibit full biological activity
Authors Mohammed Akhter Hossain, K. Johan Rosengren, Suode Zhang, Ross A. D. Bathgate, Geoffrey W. Tregear, Bianca J. van Lierop, Andrea J. Robinson and John D. Wade Published Organic & Biomolecular Chemistry Graphical abstract Abstract Replacement of disulfide bonds … Continue reading →
Controlled Synthesis of (S,S)-2,7-Diaminosuberic Acid: A Method for Regioselective Construction of Dicarba Analogues of Multicystine-Containing Peptides
Authors Jomana Elaridi, Jim Patel, W. Roy Jackson and Andrea J. Robinson Published Journal of Organic Chemistry Graphical abstract Abstract A method to facilitate regioselective formation of multiple dicarba isosteres of cystine is described. A sequence of ruthenium-catalyzed cross … Continue reading →
Dicarba α‐Conotoxin Vc1.1 Analogues with Differential Selectivity for Nicotinic Acetylcholine and GABAB Receptors
Authors Bianca J. van Lierop, Samuel D. Robinson, Shiva N. Kompella, Alessia Belgi, Jeffrey R. McArthur, Andrew Hung, Christopher A. MacRaild, David J. Adams, Raymond S. Norton and Andrea J. Robinson Published ACS Chemical Biology Graphical abstract Abstract Conotoxins … Continue reading →
Posted in Conotoxins, Dicarba peptides, Metathesis, Publications, Publications 2013
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